"PROCAINE" VITAMIN H3

Procaine Hydrochloride was first
synthesized in 1905 by a German chemist Albert Einhorn. He was looking for a
compound that would act as an anesthetic, would be non-toxic, free of side
effects, and would not be addictive.

Dr. Einhorn was looking for a
compound that could replace cocaine as an anesthetic. Cocaine was being used at
the time as an anesthetic. However, because cocaine was toxic, addictive, and
destructive to the central nervous system, its use was being outlawed. Dr. Einhorn was able to produce a
compound that demonstrated the properties he was looking for. This new compound
he named procaine. "Pro" means, in place of, and "caine" comes from the word
cocaine. Because of the similarity of the names and because they are both
anesthetics, there is much confusion as to the nature of procaine.

Procaine when injected into the
muscles acts as an anesthetic but when taken orally in a complexed form procaine
acts as a vitamin. Procaine HCl solutions, used as anesthetics, are trade named
Novocaine. Chemically procaine is the PABA
ester of amino alcohol DEAE. PABA (p-amino-benzoic acid) is a "B" vitamin.
DEAE, (n,n diethylaminoethanol) is biologically active precursor of the "B"
vitamin choline. (Fig. 1)

Procaine is usually used in the
form of the hydrochloride salt (procaine HCl) because it is highly
water-soluble. Procaine hydrochloride, when taken orally, enters the body by
being mainly absorbed through the villi in the small intestine.

Experiments show that the bulk of
the procaine HCl enters the bloodstream molecularly intact. In the blood stream
procaine HCl is rapidly hydrolyzed by the enzyme pseudo-cholinesterase into PABA
and DEAE the two components of the procaine molecule. These metabolites are
removed by the liver, chemically changed, and excreted in the urine.

In the late 1940's Dr. Ana Aslan a
Romanian cardiologist found that adding a small amount of benzoic acid to the
procaine solution stabilized some of the procaine enough to protect it from the
blood enzymes. This protected procaine, which Dr.
Aslan named Gerovital H3 or GH-3 was found to be very helpful in supplying PABA
and DEAE to damaged and or diseased cells. Ana Aslan named the procaine vitamin
H-3. GH-3 is listed under H-3 in the Merck index.

Procaine HCl when combined with
biologically active acids such as folic acid, biotin, ascorbic acid,
pantothenic acid, citric acid and many other acids such as amino acids etc. acts
as a vitamin or food supplement. The vitamin acids and other biologically
active acids when complexed with the procaine HCl molecule protect the procaine
from the enzymes in the blood allowing the procaine to enter the cells.

These vitamin complexes help the
cells assimilate and utilize nutrients more efficiently. These complexed
procaine compounds named Ultimate9.

Procaine HCl is broken down
rapidly by enzymes in the blood stream into PABA and DEAE. The PABA and DEAE
are rapidly conjugated and removed from the blood and excreted from the body.
Because of this procaine HCl and its breakdown products (metabolites) are unable
to get into the cells in any great quantity to produce benefits. Procaine HCl
will produce some benefits by itself, but they are very limited.

However when procaine HCl is
complexed properly the procaine HCl is protected from the action of the
enzymes in the blood and tissues this protection gives the procaine enough time
to be transferred into the cells of the body where it helps the cells to
rebuild, repair, and detoxify. This action of the procaine HCl complex is
responsible for the remarkable improvements in health that result from the use
of GH-3 and the Ultimate9.

Many companies claim to make
GH-3. Based lab testing the only GH-3 procaine HCl based products that
contain the active GH- factor or properly complexed procaine HCl are Ana Aslan's
injectable GH-3 and Ultimate9.

Some companies are totally
fraudulent in their claims quoting Ana Aslan case studies and my case studies
and research to validate their products, which contain no procaine HCl, or its
complexes. Their products contain PABA and
DMAE which they claim produce procaine in the body. This is false because
procaine contains no DMAE (dimethylaminoethanol). In fact the DMAE when it
enters the cells of the body is broken down and is oxidized producing by
products (metabolites) that are damaging and toxic to the cells (i.e.
formaldehyde and methyl alcohol). Whereas the DEAE (diethylaminoethanol) from
the procaine HCl breaks down in the cells and is oxidized producing acetyl
groups that are very valuable for producing acetylcholine and other materials
necessary for cellular health.

Other companies produce GH-3 and
similar products that contain procaine HCl and the other ingredients necessary
to make GH-3 and Ultimate9 and list them on their labels but they do not
have a valid product. They mix the dry ingredients together and tablet them or
put them in capsules without first forming the procaine complexes. Take the
example of making the candy called fudge. Fudge contains sugar, cocoa, condensed
milk, butter and a pinch of salt. If you mix all these together you have the
correct formula but you only have a gritty cocoa in canned milk with a chunk of
butter far from being Fudge. However if you cook the ingredients to the soft
ball stage and then allow it to cool, then beat it properly to the right
crystalline structure you end up with a delicious delight called
fudge.

The procaine HCl complexes must be
formed or the product won't be very effective in helping cells heal and overcome
their problems.

Effective procaine products in
tablets or capsules containing complexed procaine will show on the labels not
only the correct ingredients but they will also show the patent numbers of
the process for forming the complexes of procaine found in
Ultimate9.