PHARMACOLOGICAL PROPERTIES OF CLENBUTHEROL :

Farmakodinamika: selective beta2-adrenostimulyator, has a bronchodilator and secretolytic effect. Excites beta2-adrenoreceptors, stimulates adenylate cyclase, increases the content of cAMP in cells, which, by affecting the protein kinase system, deprives myosin of the ability to bind to actin and promotes anabolic steroids abuse relaxation of the bronchi. It inhibits the release from the mast cells of mediators that promote bronchospasm and inflammation of the bronchi. Reduces edema or stagnation in the bronchi, improves mucociliary clearance. In large doses causes tachycardia, tremor of fingers. The effect is observed 10-15 min after administration, reaches a maximum after 2-3 hours.

Pharmacokinetics: well absorbed after oral administration. Metabolized in the liver with the formation of 8 metabolites (in small amounts). It is excreted mainly by the kidneys (about 78% – unchanged). A small part is excreted with bile.

USE OF CLENBUTHEROL IN PREGNANCY AND IN THE LACTATION PERIOD:

It is necessary to avoid the use of the drug during pregnancy, especially in the first trimester, during the prenatal period and during childbirth. high doses can inhibit uterine contractions. Clenbuterol is probably excreted in breast milk. There is no data on the association of the use of the drug during breastfeeding with the risk for an infant, so use in nursing mothers is not recommended. The drug is used, if only the expected benefit as a result of treatment exceeds the potential risk for the child.

ADVERSE EFFECTS OF CLENBUTHEROL .

From the nervous system: tremor of fingers, anxiety, headache, dizziness, general weakness, insomnia, paresthesia. On the part of the digestive system: dry mouth, nausea, vomiting, gastralgia.

Allergic reactions: skin rash, hives, bronchospasm, angioedema.

Other: redness of the face, increased sweating, hypokalemia, muscle cramps, possible development of resistance and syndrome “rebound” when the drug is withdrawn.

CLENBUTHEROL – OVERDOSE: manifested by increased adverse reactions: arrhythmia, tachycardia, increased blood pressure, cardialgia, tremor of extremities. There is a danger of hypokalemia after an overdose, so it is necessary to monitor the serum potassium concentration.

CLENBUTHEROL – INTERACTION WITH OTHER MEDICINES: shows antagonism with beta-adrenoblockers. Reduces the effect of hypoglycemic agents. Increases the risk of developing intracardiac conduction disturbances with concomitant administration with MAO inhibitors and theophylline. Increases the toxicity of cardiac glycosides and the risk of arrhythmia. In combination with sympathomimetic agents, they increase the toxicity mutually.

In connection with the possibility of tremors, dizziness and weakness, the drug can adversely affect the ability to drive and work with machines, so during the period of treatment it is necessary to refrain from engaging in potentially dangerous activities that require increased concentration and speed of psychomotor reactions.

CLENBUTEROL – FORM OF ISSUE: bottles of dark glass, syrup (0,001 mg / ml), packed in a pack of instructions for use. and a spoon dosing

Using Clenbuterol 20 mcg Pills

It is important, however, to pay attention to the length of the Clenbuterol cycle, as well as to side effects and dosages. It isn’t safe to use for lengthy cycles (more than three or four weeks). If you do want to keep using it, you should pair it with Periactim or Ketotifen, since these antihistamines help to work against the negative effects of Clen.
Clenbuterol Hydrochloride 20 mcg is one of the most popular performance enhancing drugs available, and has both negative and side effects, as other drugs also do. It does offer many benefits. As Clenbuterol hydrochloride, it helps patents who experience breathing problems. Chronic breathing problems like asthma are often helped by this bronchodilator. Clenbuterol also helps with the relaxation of smooth muscles.

HOW TO USE CLENBUTEROL: Numerous athletes use Clenbuterol after steroid treatment to balance the resulting catabolic phase and thus obtain maximum strength and muscle mass. A further aspect of Clenbuterol is its distinct fatburning effect. Clenbuterol burns fat without dieting because it increases the body temperature slightly, forcing the body to burn fat for this process. Due to the higher body temperature Clenbuterol magnifies the effect of anabolic/androgenic steroids taken simultaneously, since the protein processing is increased.
CLENBUTEROL DOSAGE: Athletes usually take 100-140 mcg/day. For women 80-100 mcg/day are usually sufficient, It is important that the athlete begin by taking only one tablet on the first day and then increasing the dosage by one tablet each of the following days until the desired maximum dosage is reached. The compound is usually taken over a period of 8-10 weeks.

Its effect is expressed in a reduction of protein degradation in muscle cells, leading to an increase in muscle bulk and muscle strength. In the prescribed therapeutic doses, Clenbuterol has no influence on heart rate or arterial blood pressure, and does not affect oxygen saturation of arterial blood.”
The drug is indicated for:”
• treatment of bronchial asthma;
• complex therapy of bronchial spasm

Clenbuterol is a good fat burner. It can be used for decreasing body fat and weight loss.

Since Clenbuterol is not a hormone compound it has no side effects typical of anabolic steroids. For this reason it is also liked by women. Possible side effects of Clenbuterol include restlessness, palpitations, tremor (involuntary trembling of fingers), headache, increased perspiration, insomnia, possible muscle spasms, increased blood pressure, and nausea. Note that these side effects are of a temporary nature and usually subside after 8-10 days, despite continuation of the product.

To say that clenbuterol online use is rampant in bodybuilding right now would be an understatement. Thousands and thousands of athletes are using this drug. I personally know a number of pro football players, foreign Olympic athletes, and professional bodybuilders who are using clenbuterol. In addition, I have received feedback from at least 200 other athletes who have experimented with this novel compound. Generally, the feedback from clenbuterol users is that the drug produces dramatic body composition alterations. One Canadian strength coach compared the results he has seen in athletes using Clenbuterol to what one might experience while using a stack of Anavar and Halotestin. Within weeks of beginning Clenbuterol therapy, many athletes notice a significant strength increase and a dramatic reduction in body fat. The results that occur secondary to Clenbuterol administration seem to occur equally in men and women as well as young and old.