Customer Review

生物活性

技术信息

纯度 & 产品资料

参考文献

Upon intraperitoneal administration to NMRi mice, Etamicastat (100 mg/ kg) leads to a significant reduction of noradrenaline levels (36% control) in heart with concomitant increasing in dopamine levels (850% of control)[2].
Etamicastat (50 mg/kg) is rapidly absorbed into the systemic circulation reaching a maximum concentration at 4 h post-administration, representing 29% of total Etamicastat and quantified metabolites, using AUC0-t as a measure of systemic exposure[2].

Solvent & Solubility

In Vitro:

10 mM in DMSO

Preparing Stock Solutions

ConcentrationSolventMass

1 mg

5 mg

10 mg

1 mM

3.2118 mL

16.0591 mL

32.1182 mL

5 mM

0.6424 mL

3.2118 mL

6.4236 mL

10 mM

0.3212 mL

1.6059 mL

3.2118 mL

*Please refer to the solubility information to select the appropriate solvent.