VU 10010

Biological ActivitySelective allosteric potentiator of M4 acetylcholine receptors (EC50 values are 33 and 0.7 nM for ACh in the absence and presence of VU10010�respectively). Binds to an allosteric site on the receptor increasing affinity for ACh and coupling to G-proteins.

Technical Data

M.Wt:

345.85

Formula:

C17H16ClN3OS

Solubility:

Soluble to 100 mM in DMSO and to 10 mM in ethanol

Purity:

>99%

Storage:

Store at +4°C

CAS No:

633283-39-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

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